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依巴斯汀片功效

更新时间: 2021-04-23 02:05:25     

1、依巴斯汀对H1受体有高度的选择性,无中枢抑制作用。与特非那定相比,依巴斯汀作用强而持久。

2、依巴斯汀对组胺诱发的支气管痉挛具有保护作用,动物实验证实其保护作用是特非那定的4.5倍,阿斯米唑的2.9倍,连续用药不蓄积。其代谢产物Carebestine对组胺诱发的支气管痉挛的保护作用是原药的3倍。

3、依巴斯汀具有拮抗白三烯C4的作用,可抑制白三烯C4诱发的支气管痉挛,有抗胆碱作用。可抑制试验性喘息和鼻过敏。

关键词: 功效

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